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pp-H1

Gene
pp-H1
Protein
Phyllokinin-1
Organism
Phyllomedusa azurea
Length
62 amino acids
Function
[Thr6]-bradykinin: inhibits ACE with a Ki of 1.6 uM, and targets B2 bradykinin receptor (BDKRB2). Provokes contraction of smooth muscle preparation (ileum). In vivo, induces an early hyperalgesic effects in living rats after intraplantar injection (By similarity).
Similarity
Belongs to the bradykinin-related peptide family.
Mass
7.386 kDa
Sequence
MSFLKKSLFLVLFLGLVSSSICEEEKRETEEEENEDEIEEESEEKKREDPERPPGFTPFRVY